Staff Profile
Professor David Fulton
- Address: Chemistry
School of Natural and Environmental Sciences
Bedson Building (3.44)
Newcastle University
Newcastle upon Tyne
NE1 7RU
Background
Biography
David Fulton received his BSc (Hons) from Strathclyde University and PhD from the University of California, Los Angeles, working on carbohydrate and supramolecular chemistry under the direction of Prof Sir J Fraser Stoddart FRS. He then spent two and half years as a postdoctoral research associate with Prof David Parker FRS at the University of Durham working on the synthesis of gadolinium-centered dendrimers as new MRI contrast agents. In 2006 he moved up the road to take up his present position within Chemistry at Newcastle University where he is a member of its Functional Materials and Molecules group. His research interests are broadly based upon supramolecular/synthetic polymer chemistry.
Qualifications
PhD University of California, Los Angeles, 2001
BSc (Hons) University of Strathclyde, 1996
Previous Positions
Postdoctoral Research Associate, Durham University, 2003-2005
Analytical Method Development Chemist, Quintiles Ltd, 2002
Process Development Chemist, Merck Ltd, 1994-1995
Area of Expertise
Supramolecular polymers and materials.
Google Scholar
https://scholar.google.co.uk/citations?user=NDGx0nAAAAAJ&hl=en
Research
Dr David Fulton has broad interests in polymer and supramolecular chemistry. Projects have received support from EPSRC, Innovate UK, The EU-framework 7 program, industrial partners and The Royal Society. Some current projects are summarized.
Polymers and materials from bacterial fimbriae. For millennia, humans have exploited fibres produced by animals and plants to make materials such as textiles and paper. Many strains of bacteria also produce hair-like fibres called fimbriae that have evolved unique structural and mechanical properties that make them appealing building as the foundation for new materials, however, these possibilities are still essentially unexplored.
Working closely with the laboratory of Prof Jeremy Lakey at Newcastle, we have developed the first examples of materials based upon Capsular antigen fragment 1 (Caf1) (Fig. 1a), the fimbriae produced in nature by Yersinia Pestis, the bacterium responsible for the bubonic plague.
Caf1 polymers (~ 1 µm) are chains of 15 kDa monomer subunits, each non-covalently linked to a single neighbouring subunit by a donated N-terminal β-strand. Caf1 has evolved its structure to inhibit interactions with host cells, helping the bacterium hide from the immune system. Caf1 bears a structural resemblance to fibronectin—a naturally occurring extracellular matrix—suggest Caf1 has great potential as a biomaterial for advanced cell culture. It is possible to ‘hard-wire’ cell adhesion peptides into surface loops of the Caf1 protein, presenting a straightforward way to engineer bioactivity whilst avoiding chemical functionalization with expensive peptides. This structural similarity to ECM proteins, together with its other highly desirable properties (non-adhesion, stability and ease of production) endow Caf1 with features that are difficult to design de novo into protein polymers. Furthermore, Caf1 is produced by bacterial fermentation and thus does not suffer from the batch-to-batch variability of animal-based materials such as Matrigel®.
It is easy to chemically cross-link Caf1 polymers into hydrogel materials (Fig. 2a,b), 3D polymer networks possessing high water contents and porous structures, properties they share with the extracellular matrix.
Caf1 also has some hidden and unexpected features. The linkages between subunits in the Caf1 are exceptionally strong and kinetically very inert, however, we discovered that heat can be used to reversibly cycle Caf1 between its polymeric and monomeric states (Fig. 3), a feature that endows the Caf1 polymer with new synthetic and materials possibilities. This has allowed us to prepare copolymers featuring controlled compositions of naturally-occurring and mutant subunits, and to encapsulate live cells within a cross-linked Caf1 matrix.
Dynamic Covalent Polymers. Dynamic covalent chemistry relates to chemical reactions carried out under conditions of equilibrium control, and exploits dynamic covalent bonds (DCBs), which like non-covalent bonds display a dynamic nature but which also possess the chemical robustness associated with all covalent bonds. The term ‘dynamic covalent bond’ simply describes any covalent chemical bond which possesses the capacity to be formed and broken under equilibrium control, and encompasses many well-known functional groups such as imines, esters and hydrazone. At Newcastle we have been utilizing DCBs to endow polymeric systems with the abilities to adapt their structures or compositions in response to an external stimuli. When DCBs are incorporated into polymeric systems, the reversible nature of bonds enables these systems to modify their architectures by reshuffling, incorporating or releasing their components, in effect providing a mechanism for polymer systems to reconfigure their molecular structures and therefore their functional or material properties.
One way we have utilized these ideas is in the development of polymer-scaffolded dynamic combinatorial libraries which we have shown respond to the addition of macromolecular templates by changing their compositions, preferentially incorporating residues which promote binding and rejecting residues which do not. This work might lead to a new method to make artificial receptors for sensing and separations.
We have also developed dynamic covalent polymers which are able to undergo structural metamorphosis from an intramolecularly cross-linked polymer chain into cross-linked gels or films, and we are working to develop this approach to allow the ‘wrapping’ of small biological objects such as viruses or bacteria within cross-linked polymer films.
Polymers for Industrial Applications. Polymers have been a component of detergent/cleaner formulations for many years, where their purpose is to improve product performance. Many of these polymers, however, are petrochemical-based with worldwide consumption > 130,000 tonnes p/a. Concerns regarding depletion of fossil resources, disposal and related issues, as well as evolving government policies, are driving the search for alternatives, and there is now an urgent need to develop bio-based and biodegradable alternatives to petrochemical-based polymers. Polysaccharides are of considerable potential as they are usually derived from sustainable plant sources and are associated with low toxicity and excellent biodegradability. We are working in collaboration with Procter & Gamble to develop new polysaccharide biopolymers derived from sustainable feedstocks that create novel functionalities including polymers that entrap hydrophobic guests within their 3D structures (potential for dye transfer inhibition, hydrophobic soil suspension) and as flexible amphiphilic polymers (beneficial for anti-redeposition).
The fouling of surfaces by marine organisms presents a substantial problem, leading to reduced vessel performance and increased costs. Traditional solutions have involved antifouling coatings which leach biocides (often based upon tin or copper) but because of the adverse impact caused by the release of toxic compounds into the environment these coatings are either banned or under increasing regulatory scrutiny. Working with Akzo Nobel and Solvay, we have developed zwitterionic foul-release polymer coatings which display potential in marine antifouling applications.
Teaching
Undergraduate Teaching
Stage 2 Organic chemistry (NES2402): Module leader and lecturer (22 lectures).
Stage 3 Organic chemistry (NES3402): Lecturer (11 lectures).
Stage 3 Analytical Chemistry (NES341): Module leader
I also contribute to a number of other modules including final year MChem project supervision( CHY8511) and MSc project supervision (NES8002).
Publications
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Articles
- Leung CCH, Dura G, Waller H, Lakey JH, Fulton DA. The encapsulation and controlled release of proteins from “meltable” chemically cross-linked hydrogels. Journal of Applied Polymer Science 2024, epub ahead of print.
- D'Avino M, Chilton R, Si G, Sivik MR, Fulton DA. Pullulan Derivatives as Softening and Cleaning Additives for Laundry Detergents. Industrial and Engineering Chemistry Research 2023, 62(51), 21909-21917.
- Upson SJ, Benning MJ, Fulton DA, Corbett IP, Dalgarno KW, German MJ. Bond Strength and Adhesion Mechanisms of Novel Bone Adhesives. Bioengineering 2023, 10(1), 78.
- Banks AM, Whitfield CJ, Brown SR, Fulton DA, Goodchild SA, Grant C, Love J, Lendrem D, Fieldsend JE, Howard TP. Key reaction components affect the kinetics and performance robustness of cell-free protein synthesis reactions. Computational and Structural Biotechnology Journal 2022, 20, 218-229.
- Dura G, Crespo-Cuadrado M, Waller H, Peters DT, Ferreira-Duarte A, Lakey JH, Fulton DA. Exploiting Meltable Protein Hydrogels to Encapsulate and Culture Cells in 3D. Macromolecular Bioscience 2022, 22(9), 2200134.
- D'Avino M, Chilton R, Gang S, Sivik MR, Fulton DA. Evaluating the Role of Hydrophobic and Cationic Appendages on the Laundry Performance of Modified Hydroxyethyl Celluloses. Industrial and Engineering Chemistry Research 2022, 61(38), 14159-14172.
- Solovyova AS, Peters DT, Dura G, Waller H, Lakey JH, Fulton DA. Probing the oligomeric re-assembling of bacterial fimbriae in vitro: a small-angle X-ray scattering and analytical ultracentrifugation study. European Biophysics Journal 2021, 50, 597-611.
- Dura G, Crespo-Cuadrado M, Waller H, Peters DT, Ferreira AM, Lakey JH, Fulton DA. Hydrogels of engineered bacterial fimbriae can finely tune 2D human cell culture. Biomaterials Science 2021, 9(7), 2542-2552.
- Feng Z, Esteban PO, Gupta G, Fulton DA, Mamlouk M. Highly conductive partially cross-linked poly(2,6-dimethyl-1,4-phenylene oxide) as anion exchange membrane and ionomer for water electrolysis. International Journal of Hydrogen Energy 2021, 46(75), 37137-37151.
- Higgs PL, Appleton JL, Turnbull WB, Fulton DA. Exploiting the Structural Metamorphosis of Polymers to 'Wrap' Micron-Sized Spherical Objects. Chemistry - A European Journal 2021, 27(70), 17647-17654.
- Ruiz-Sanchez AJ, Guerin AJ, El-Zubir O, Dura G, Ventura C, Dixon LI, Houlton A, Horrocks BR, Jakubovics NS, Guarda P-A, Simeone G, Clare AS, Fulton DA. Preparation and evaluation of fouling-release properties of amphiphilic perfluoropolyether-zwitterion cross-linked polymer films. Progress in Organic Coatings 2020, 140, 105524.
- Whitfield CJ, Banks AM, Dura G, Love J, Fieldsend JE, Goodchild SA, Fulton DA, Howard TP. Cell-free protein synthesis in hydrogel materials. Chemical Communications 2020, 56(52), 7108-7111.
- Dura G, Peters DT, Waller H, Yemm AI, Perkins ND, Ferreira AM, Crespo-Cuadrado M, Lakey JH, Fulton DA. A thermally reformable protein polymer. Chem 2020, 6(11), 3132-3151.
- Bracchi ME, Dura G, Fulton DA. The synthesis of poly(arylthiols) and their utilization in the preparation of cross-linked dynamic covalent polymer nanoparticles and hydrogels. Polymer Chemistry 2019, 10(10), 1258-1267.
- Higgs PL, Ruiz-Sanchez AJ, Dalmina M, Horrocks BR, Leach AG, Fulton DA. Enhancing the kinetics of hydrazone exchange processes: An experimental and computational study. Organic and Biomolecular Chemistry 2019, 17(12), 3218-3224.
- Dura G, Waller H, Gentile P, Lakey JH, Fulton DA. Tuneable hydrogels of Caf1 protein fibers. Materials Science and Engineering C 2018, 93, 88-95.
- Ulusu Y, Dura G, Waller H, Benning MJ, Fulton DA, Lakey JH, Peters DH. Thermal stability and rheological properties of the ‘non-stick’ Caf1 biomaterial. Biomedical Materials 2017, 12(5), 051001.
- Ruiz-Sanchez AJ, Higgs PL, Peters DT, Turley AT, Dobson MA, North AJ, Fulton DA. Probing the Surfaces of Biomacromolecules with Polymer-Scaffolded Dynamic Combinatorial Libraries. ACS Macro Letters 2017, 6(9), 903-907.
- Borah D, Cummins C, Rasappa S, Watson SMD, Pike AR, Horrocks BR, Fulton DA, Houlton A, Liontos G, Ntetsikas K, Avgeropoulos A, Morris MA. Nanoscale silicon substrate patterns from self-assembly of cylinder forming poly (styrene)-block-poly(dimethylsiloxane) block copolymer on silane functionalized surfaces. Nanotechnology 2017, 28(4).
- Mahon CS, McGurk CJ, Watson SMD, Fascione MA, Sakonsinsiri C, Turnbull WB, Fulton DA. Molecular recognition-mediated transformation of single-chain polymer nanoparticles into crosslinked polymer films. Angewandte Chemie International Edition 2017, 56(42), 12913-12918.
- Ventura C, Guerin AJ, El-Zubir O, Ruiz-Sanchez AJ, Dixon LI, Reynolds KJ, Dale ML, Ferguson J, Houlton A, Horrocks BR, Clare AS, Fulton DF. Marine antifouling performance of polymer coatings incorporating zwitterions. Biofouling 2017, 33(10), 892-903.
- Upson SJ, Partridge SW, Tcacencu I, Fulton DA, Corbett I, German MJ, Dalgarno KW. Development of a methacrylate-terminated PLGA copolymer for potential use in craniomaxillofacial fracture plates. Materials Science and Engineering C 2016, 69, 470-477.
- Mahon CS, Fascione MA, Sakonsinsiri CS, McAllister TE, Turnbull WB, Fulton DA. Templating carbohydrate-functionalised polymer-scaffolded dynamic combinatorial libraries with lectins. Organic & Biomolecular Chemistry 2015, 13(9), 2756-2761.
- Bracchi ME, Fulton DA. Orthogonal breaking and forming of dynamic covalent imine and disulfide bonds in aqueous solution. Chemical Communications 2015, 51(55), 11052-11055.
- Sanchez-Sanchez A, Fulton DA, Pomposo JA. pH-responsive single-chain polymer nanoparticles utilising dynamic covalent enamine bonds. Chemical Communications 2014, 50(15), 1871-1874.
- Harun NA, Horrocks BR, Fulton DA. Enhanced Raman and luminescence spectra from co-encapsulated silicon quantum dots and Au-Ag nanoalloys. Chemical Communications 2014, 50(82), 12389-12391.
- Whitaker DE, Mahon CS, Fulton DA. Thermoresponsive Dynamic Covalent Single-Chain Polymer Nanoparticles Reversibly Transform into a Hydrogel. Angewandte Chemie: International Edition 2013, 52(3), 956-959.
- Mahon CS, Fulton DA. Templation-induced re-equilibration in polymer-scaffolded dynamic combinatorial libraries leads to enhancements in binding affinities. Chemical Science 2013, 4, 3661-3666.
- Mahon CS, Jackson AW, Murray BS, Fulton DA. Investigating templating within Polymer-Scaffolded Dynamic Combinatorial Libraries. Polymer Chemistry 2013, 4, 368–377.
- Harun NA, Benning MJ, Horrocks BR, Fulton DA. Gold nanoparticle-enhanced luminescence of silicon quantum dots co-encapsulated in polymer nanoparticles. Nanoscale 2013, 5(9), 3817-3827.
- Omedes Pujol M, Coleman DJL, Allen CD, Heidenreich O, Fulton DA. Determination of key structure-activity relationships in siRNA delivery with a mixed micelle system. Journal of Controlled Release 2013, 172(3), 939-945.
- Jackson AW, Fulton DA. Triggering Polymeric Nanoparticle Disassembly Through the Simultaneous Application of Two Different Stimuli. Macromolecules 2012, 45(6), 2699-2708.
- Jackson AW, Stakes C, Fulton DA. The formation of core cross-linked star polymer and nanogel assemblies facilitated by the formation of dynamic covalent imine bonds. Polymer Chemistry 2011, 2(11), 2500-2511.
- Mahon CS, Jackson AW, Murray BS, Fulton DA. Templating a polymer-scaffolded dynamic combinatorial library. Chemical Communications 2011, 47(25), 7209-7211.
- Jackson AW, Fulton DA. pH triggered self-assembly of core cross-linked star polymers possessing thermoresponsive cores. Chemical Communications 2011, 47(24), 6807-6809.
- Murray BS, Fulton DA. Dynamic Covalent Single-Chain Polymer Nanoparticles. Macromolecules 2011, 44(18), 7242-7252.
- Harun NA, Horrocks BR, Fulton DA. A miniemulsion polymerization technique for encapsulation of silicon quantum dots in polymer nanoparticles. Nanoscale 2011, 3(11), 4733-4741.
- Jackson AW, Fulton DA. The formation of core cross-linked star polymers containing cores cross-linked by dynamic covalent imine bonds. Chemical Communications 2010, 46(33), 6051-6053.
- Murray BS, Jackson AW, Mahon CS, Fulton DA. Reactive Thermoresponsive Copolymer Scaffolds. Chemical Communications 2010, 46, 8651-8653.
- Jackson AW, Fulton DA. Dynamic Covalent Diblock Copolymers Prepared from RAFT Generated Aldehyde and Alkoxyamine End-Functionalized Polymers. Macromolecules 2010, 43(2), 1069-1075.
- Fulton DA. Dynamic combinatorial libraries constructed on polymer scaffolds. Organic Letters 2008, 10(15), 3291-3294.
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Note
- Fulton DA. Synthesis: Click chemistry gets reversible. Nature Chemistry 2016, 8(10), 899-900.
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Reviews
- Fulton DA, Dura G, Peters DT. The polymer and materials science of the bacterial fimbriae Caf1. Biomaterials Science 2023, 22(11), 7229-7246.
- Mahon CS, Fulton DA. Mimicking nature with synthetic macromolecules capable of recognition. Nature Chemistry 2014, 6(8), 665-672.
- Jackson AW, Fulton DA. Making polymeric nanoparticles stimuli-responsive with dynamic covalent bonds. Polymer Chemistry 2013, 4(1), 31-45.